Examining Methyl-1-Testosterone: The Potent Underground Oral Steroid

Assessing Its Reputation, Toxicity, and Legal Status

Background and History

Methyl-1-Testosterone, also known as 17α-methyl-δ1-dihydroboldenone or methyldihydroboldenone, is a modified form of the steroid boldenone. It was first developed in the 1960s but was never approved for human use. It began appearing on the black market used almost exclusively by bodybuilders and athletes.

Methyl-1-Testosterone gained a reputation as a powerful oral steroid for building muscle and strength, but also came with considerable side effects. Supply was also scarce, limiting its widespread use. Today it remains available primarily through underground labs and networks.

Chemical Structure

The chemical structure of Methyl-1-Testosterone consists of boldenone with an added 17-alpha-methyl group to enable oral administration. It also contains a double bond between carbons 1 and 2. The modifications greatly enhance its anabolic strength.

Dosages and Cycles

Effective doses of Methyl-1-Testosterone are 15-30mg daily, taken orally for 4-6 weeks on average. The relatively short cycles and low doses help mitigate toxicity issues. Stacking with injectable steroids is common practice.

Effects and Benefits

Methyl-1-Testosterone is valued for providing significant gains in muscle hypertrophy, lean mass, and strength. It also enhances collagen synthesis and bone strength. The methylation makes it resistant to aromatization and conversion to DHT.

Side Effects and Health Risks

However, methyl-1-testosterone can produce harsh side effects:

• • Hepatotoxicity and potential liver damage

• • LDL/HDL cholesterol imbalances

• • High blood pressure

• • Testosterone suppression

• • Negative cardiovascular effects

This makes cycling, dosing, and stacks critical for moderating side effects. Short cycles and prudent dosing is advised. It also must be avoided if pre-existing health conditions are present.

Legal Status

In the United States, methyl-1-testosterone is classified as a Schedule III controlled substance under federal regulation. It is only legal to possess and use with a valid prescription, which is extremely rare. Underground manufacturing and black market trade continues to defy prohibition.

In summary, methyl-1-testosterone is a uniquely potent oral steroid, but its toxicity and legal status warrants caution by any prospective user. Safer legal supplements exist today providing comparable benefits.